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NAN-190 hydrobromide

CAS No. 115338-32-4

NAN-190 hydrobromide ( NAN190 hydrobromide;NAN 190 hydrobromide )

产品货号. M10539 CAS No. 115338-32-4

NAN-190 is a 5-HT1A receptor antagonist with Ki of 0.6 nM; also potently blocks the α2-adrenergic receptor.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥259 有现货
10MG ¥373 有现货
50MG ¥599 有现货
100MG ¥778 有现货
200MG ¥1401 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    NAN-190 hydrobromide
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    NAN-190 is a 5-HT1A receptor antagonist with Ki of 0.6 nM; also potently blocks the α2-adrenergic receptor.
  • 产品描述
    NAN-190 is a 5-HT1A receptor antagonist with Ki of 0.6 nM; also potently blocks the α2-adrenergic receptor; antagonizes the stimulation by norepinephrine of phosphoinositide turnover in rat cortical slices.Anxiety Preclinical
  • 同义词
    NAN190 hydrobromide;NAN 190 hydrobromide
  • 通路
    Endocrinology/Hormones
  • 靶点
    5-HT Receptor
  • 受体
    5-HT Receptor
  • 研究领域
    Neurological Disease
  • 适应症
    Anxiety

化学信息

  • CAS Number
    115338-32-4
  • 分子量
    474.39
  • 分子式
    C23H28BrN3O3
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO: 36.23 mg/mL
  • SMILES
    COC1=CC=CC=C1N2CCN(CC2)CCCCN3C(=O)C4=CC=CC=C4C3=O.Br
  • 化学全称
    1H-Isoindole-1,3(2H)-dione, 2-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-, hydrobromide (1:1)

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Claustre Y, et al. Eur J Pharmacol. 1991 Oct 29;204(1):71-7.
2. Zhang J, et al. J Neurosci. 2010 Feb 17;30(7):2433-41.
3. Glennon RA, et al. J Med Chem. 1988 Oct;31(10):1968-71.
产品手册
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